Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Phosphatase Inhibitor Cocktail Set III
Phosphatase Inhibitor Cocktail Set III is a ready to use cocktail of four phosphatase inhibitors for broad-spectrum inhibition of both serine/threonine and protein tyrosine phosphatases.
MilliporeSigma™ Calbiochem™ NG,NG-Dimethyl-L-arginine, Dihydrochloride
A cell-permeable, reversible inhibitor of nitric oxide synthase in vitro (IC50 = 2-3 μM) and in vivo.
MilliporeSigma™ Calbiochem™ 17-DMAG
A potent antitumor analog of 17-AAG that binds to the ATPase site of human Hsp90α with high affinity and displays excellent bioavailability and aqueous solubility.
MilliporeSigma™ Calbiochem™ SIRT1 Activator II
The SIRT1 Activator II, also referenced under CAS 374922-43-7, modulates the biological activity of SIRT1. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ InSolution™ PKR Inhibitor
The InSolution™ PKR Inhibitor, also referenced under CAS 608512-97-6, controls the biological activity of PKR. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ NFAT Inhibitor, Cell-Permeable
The NFAT Inhibitor, Cell-Permeable controls the biological activity of NFAT. This small molecule/inhibitor is primarily used for Inflammation/Immunology applications.
MilliporeSigma™ Calbiochem™ CDC42 Inhibitor III, ZCL278
A cell-permeable, non-cytotoxic, aqueous soluble (181μM in PBS, pH 7
MilliporeSigma™ Calbiochem™ JNK Inhibitor IX
The JNK Inhibitor IX, also referenced under CAS 312917-14-9, controls the biological activity of JNK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ CGP 37849
A highly potent competitive antagonist selective for NMDA receptors (Ki = 35
MilliporeSigma™ Calbiochem™ MMP-2/MMP-3 Inhibitor III, PD166793
The MMP-2/MMP-3 Inhibitor III, PD166793, also referenced under CAS 199850-67-4, controls the biological activity of MMP-2/MMP-3. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ InSolution™ Jasplakinolide, Jaspis johnstoni
InSolution™ Jasplakinolide, Jaspis johnstoni, CAS 102396-24-7, is a 1mm solution of Jasplakinolide, Jaspis johnstoni in DMSO. Acts as a potent inducer of actin polymerization and stabilization.
MilliporeSigma™ Calbiochem™ Adenosine A1 Receptor Antagonist I, DPCPX
A blood-brain barrier permeable xanthine derivative that acts as a highly selective antagonist of Adenosine A1 receptor (A1R; Ki
MilliporeSigma™ Calbiochem™ Mer RTK Inhibitor, UNC569
The Mer RTK Inhibitor, UNC569 controls the biological activity of Mer RTK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ AdaAhx3L3VS
A potent, covalent, cell-permeable, irreversible inhibitor of chymotrypsin-like (50-100 nM), trypsin-like (1-5 μM), and PGPH (0.5-1 μM) activities of the 20S proteasome.
MilliporeSigma™ Calbiochem™ Transglutaminase 2 Inhibitor, ZDON
A cell-permeable, peptide-based, irreversible inhibitor of transglutaminase 2 (TG2; IC50 = 150nM for recombinant TG2). Reacts with the active site cysteine of TG2.